发明名称 |
PROCESS FOR THE PREPARATION OF OPTICALLY ACTIVE (S)-(+)-N,N-DIMETHYL-3-(1-NAPHTHALENYLOXY)-3-(2-THIENYL)PROPANAMINE |
摘要 |
<p>Diasteromerically enriched salts Of (S)-DNTH<SUP>+</SUP> EPA<SUP>-</SUP> and (R)-DNTH<SUP>+</SUP> EPA<SUP>-</SUP>, methods of preparing such diasteromerically enriched salts Of (S)-DNTH<SUP>+</SUP> EPA<SUP>-</SUP> and (R)-DNTH<SUP>+ </SUP>EPA<SUP>-</SUP>, and methods of preparing enantiomerically enriched (S)-DNT and enantiomerically enriched (R)-DNT are provided.</p> |
申请公布号 |
WO2006099459(A1) |
申请公布日期 |
2006.09.21 |
申请号 |
WO2006US09247 |
申请日期 |
2006.03.14 |
申请人 |
TEVA PHARMACEUTICAL INDUSTRIES LTD.;TEVA PHARAMCEUTICAL USA, INC.;INI, SANTIAGO;ABRAMOV, MILI;LIBERMAN, ANITA |
发明人 |
INI, SANTIAGO;ABRAMOV, MILI;LIBERMAN, ANITA |
分类号 |
C07D233/22;A61K31/38;A61P13/00;A61P25/24;A61P29/00 |
主分类号 |
C07D233/22 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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