发明名称 PEPTIDASE INHIBITORS
摘要 The present invention relates to a series of novel compounds having the formula (I) wherein: X is NR<SUP>3</SUP> or O; n is 1 or 2; A is a bicyclic carbocycle and R1 and R2 are as described herein. The compounds are useful as DPP-IV inhibitors, such as for the treatment of diabetes.
申请公布号 WO2006012395(A3) 申请公布日期 2006.05.04
申请号 WO2005US25837 申请日期 2005.07.21
申请人 ROYALTY, SUSAN MARIE;BURNS, JAMES FORD;SCICINSKI, JAN JOZEF;JAGDMANN, JR., GUNNAR ERIK;FOGLESONG, ROBERT JAMES;GRIFFIN, KELLEE RENEE;DYAKONOV, TATYANA;MIDDLEMISS, DAVID 发明人 ROYALTY, SUSAN MARIE;BURNS, JAMES FORD;SCICINSKI, JAN JOZEF;JAGDMANN, JR., GUNNAR ERIK;FOGLESONG, ROBERT JAMES;GRIFFIN, KELLEE RENEE;DYAKONOV, TATYANA;MIDDLEMISS, DAVID
分类号 C07D207/09;A61K31/4025;C07D207/10 主分类号 C07D207/09
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