发明名称 METHOD OF SYNTHESISING (1S)-4,5-DIMETHOXY-1- (METHYLAMINOMETHYL)-BENZOCYCLOBUTANE AND THE ADDITION SALTS THEREOF, AND USE OF SAME FOR THE SYNTHESIS OF IVABRADINE AND THE PHARMACEUTICALLY-ACCEPTABLE ADDITION SALTS THEREOF
摘要 <p>The invention relates to a method of synthesising a compound having formula (I) and to the use thereof for the synthesis of ivabradine and the pharmaceutically-acceptable acid addition salts and hydrates of same.</p>
申请公布号 WO2005123659(A1) 申请公布日期 2005.12.29
申请号 WO2005FR00397 申请日期 2005.02.21
申请人 LES LABORATOIRES SERVIER;LERESTIF, JEAN-MICHEL;GONZALES BLANCO, ISAAC;LECOUVE, JEAN-PIERRE;BRIGOT, DANIEL 发明人 LERESTIF, JEAN-MICHEL;GONZALES BLANCO, ISAAC;LECOUVE, JEAN-PIERRE;BRIGOT, DANIEL
分类号 C07D223/16;A61K31/55;A61P9/06;A61P9/10;C07B57/00;C07B61/00;C07C213/02;C07C213/08;C07C213/10;C07C217/56;C07C217/58;(IPC1-7):C07C213/10 主分类号 C07D223/16
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