发明名称 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions and uses thereof
摘要 Compounds of Formula (I) wherein R<SUP>1</SUP>, R<SUP>2</SUP>, R<SUP>3</SUP>, R<SUP>4</SUP>, R<SUP>5</SUP>, R<SUP>6 </SUP>and X are as defined herein for Formula (IA) and Formula (IB), or a tautomer, prodrug, solvate, or salt thereof; pharmaceutical compositions containing such compounds, and methods of modulating the glucocorticoid receptor function and methods of treating disease-states or conditions mediated by the glucocorticoid receptor function or characterized by inflammatory, allergic, or proliferative processes in a patient using these compounds.
申请公布号 US2005234091(A1) 申请公布日期 2005.10.20
申请号 US20050072819 申请日期 2005.03.04
申请人 BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. 发明人 REGAN JOHN R.;LEE THOMAS W.;THOMSON DAVID;KIRRANE THOMAS M.JR.;KUZMICH DANIEL;PROUDFOOT JOHN R.;BEKKALI YOUNES;ZINDELL RENEE
分类号 A61K31/4355;A61K31/4365;A61K31/437;A61K31/4375;A61K31/4741;A61K31/4743;A61K31/4745;C07D471/02;C07D471/04;C07D491/02;C07D491/04;C07D495/04;C07D498/02;C07D498/04;C07D513/04;(IPC1-7):C07D471/02;A61K31/474 主分类号 A61K31/4355
代理机构 代理人
主权项
地址