发明名称 |
NOVEL COMPOUNDS AND COMPOSITIONS AS CATHEPSIN INHIBITORS |
摘要 |
The present invention relates to novel selective cathepsin S inhibitors, the pharmaceutically acceptable salts and N-oxides thereof, their uses as therapeutic agents and the methods of their making. |
申请公布号 |
HRP20030995(A2) |
申请公布日期 |
2005.08.31 |
申请号 |
HR2003P000995 |
申请日期 |
2003.11.28 |
申请人 |
AVENTIS PHARMACEUTICALS INC. AXYS PHARMACEUTICALS |
发明人 |
MICHAEL GRAUPE;JIAYAO LI;LINK JOHN;SHEILA ZIPFEL;TIMM PAUL ANDREAS;ALDOUS JOHN DAVID;SUKANTHINI THURAIRATNAM |
分类号 |
C07D295/18;A61K31/165;A61K31/277;A61K31/341;A61K31/351;A61K31/381;A61K31/397;A61K31/40;A61K31/423;A61K31/4245;A61K31/426;A61K31/427;A61K31/428;A61K31/437;A61K31/4453;A61K31/4468;A61K31/454;A61K31/495;A61K31/5375;A61K31/5377;A61K31/55;A61P1/02;A61P13/12;A61P19/02;A61P21/04;A61P29/00;A61P33/06;A61P35/00;A61P43/00;C07C233/31;C07C255/29;C07C255/44;C07C255/46;C07C271/12;C07C271/16;C07C271/22;C07C271/24;C07C317/44;C07C317/46;C07C317/48;C07D205/04;C07D207/08;C07D207/16;C07D211/66;C07D223/08;C07D223/12;C07D239/08;C07D263/56;C07D271/06;C07D271/10;C07D277/28;C07D277/64;C07D277/82;C07D295/185;C07D295/20;C07D295/205;C07D307/14;C07D309/14;C07D333/24;C07D413/12;C07D413/14;C07D417/12;C07D498/04 |
主分类号 |
C07D295/18 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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