发明名称 Antithrombotic agents
摘要 This application relates to a compound of formula I (or a prodrug thereof or a pharmaceutically acceptable salt of the compound or prodrug thereof) as defined herein, pharmaceutical compositions thereof, and its use as an inhibitor of factor Xa, as well as a process for its preparation and intermediates therefor.
申请公布号 US2003195223(A1) 申请公布日期 2003.10.16
申请号 US20020133907 申请日期 2002.04.25
申请人 BEIGHT DOUGLAS WADE;CRAFT TRELIA JOYCE;FRANCISKOVICH JEFFRY BERNARD;GOODSON THEODORE;HALL STEVEN EDWARD;HERRON DAVID KENT;KLIMKOWSKI VALENTINE JOSEPH;MASTERS JOHN JOSEPH;MENDEL DAVID;MILOT GUY;SAWYER JASON SCOTT;SHUMAN ROBERT THEODORE;SMITH GERALD FLOYD;TEBBE ANNE LOUISE;TINSLEY JENNIFER MARIE;WEIR LEONARD CRAYTON;WIKEL JAMES HOWARD;WILEY MICHAEL ROBERT;YEE YING KWONG 发明人 BEIGHT DOUGLAS WADE;CRAFT TRELIA JOYCE;FRANCISKOVICH JEFFRY BERNARD;GOODSON THEODORE;HALL STEVEN EDWARD;HERRON DAVID KENT;KLIMKOWSKI VALENTINE JOSEPH;MASTERS JOHN JOSEPH;MENDEL DAVID;MILOT GUY;SAWYER JASON SCOTT;SHUMAN ROBERT THEODORE;SMITH GERALD FLOYD;TEBBE ANNE LOUISE;TINSLEY JENNIFER MARIE;WEIR LEONARD CRAYTON;WIKEL JAMES HOWARD;WILEY MICHAEL ROBERT;YEE YING KWONG
分类号 C07D333/40;A61K31/00;A61K31/167;A61K31/196;A61K31/216;A61K31/27;A61K31/381;A61K31/4035;A61K31/423;A61K31/445;A61K31/4545;A61P7/02;C07C257/18;C07C259/18;C07C271/64;C07C271/66;C07D209/44;C07D211/60;C07D261/20;C07D333/38;C07D401/04;(IPC1-7):A61K31/435;A61K31/325;A61K31/195 主分类号 C07D333/40
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