发明名称 |
Antithrombotic agents |
摘要 |
This application relates to a compound of formula I (or a prodrug thereof or a pharmaceutically acceptable salt of the compound or prodrug thereof) as defined herein, pharmaceutical compositions thereof, and its use as an inhibitor of factor Xa, as well as a process for its preparation and intermediates therefor.
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申请公布号 |
US2003195223(A1) |
申请公布日期 |
2003.10.16 |
申请号 |
US20020133907 |
申请日期 |
2002.04.25 |
申请人 |
BEIGHT DOUGLAS WADE;CRAFT TRELIA JOYCE;FRANCISKOVICH JEFFRY BERNARD;GOODSON THEODORE;HALL STEVEN EDWARD;HERRON DAVID KENT;KLIMKOWSKI VALENTINE JOSEPH;MASTERS JOHN JOSEPH;MENDEL DAVID;MILOT GUY;SAWYER JASON SCOTT;SHUMAN ROBERT THEODORE;SMITH GERALD FLOYD;TEBBE ANNE LOUISE;TINSLEY JENNIFER MARIE;WEIR LEONARD CRAYTON;WIKEL JAMES HOWARD;WILEY MICHAEL ROBERT;YEE YING KWONG |
发明人 |
BEIGHT DOUGLAS WADE;CRAFT TRELIA JOYCE;FRANCISKOVICH JEFFRY BERNARD;GOODSON THEODORE;HALL STEVEN EDWARD;HERRON DAVID KENT;KLIMKOWSKI VALENTINE JOSEPH;MASTERS JOHN JOSEPH;MENDEL DAVID;MILOT GUY;SAWYER JASON SCOTT;SHUMAN ROBERT THEODORE;SMITH GERALD FLOYD;TEBBE ANNE LOUISE;TINSLEY JENNIFER MARIE;WEIR LEONARD CRAYTON;WIKEL JAMES HOWARD;WILEY MICHAEL ROBERT;YEE YING KWONG |
分类号 |
C07D333/40;A61K31/00;A61K31/167;A61K31/196;A61K31/216;A61K31/27;A61K31/381;A61K31/4035;A61K31/423;A61K31/445;A61K31/4545;A61P7/02;C07C257/18;C07C259/18;C07C271/64;C07C271/66;C07D209/44;C07D211/60;C07D261/20;C07D333/38;C07D401/04;(IPC1-7):A61K31/435;A61K31/325;A61K31/195 |
主分类号 |
C07D333/40 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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