发明名称 |
COMPOUNDS ACTING AS MELANOCORTIN RECEPTOR LIGANDS |
摘要 |
The present invention provides novel compounds and use of compounds of gener al formula (I) as ligands to the melanocortin receptors and/or for treatment of disorders in the melanocortin system: Wherein X and Y are independently chos en from O, N, S and (CH2)n, where n is 0, 1, 2, 3, 4 or 5, or a combination of these and may contain carbon-carbon multiple bonds and branched chains as we ll as alicyclic and heterocyclic groups; Q is H or OH; R1 and R2 can be either the same or different and are chosen from hydrogen or the residue of an aromatic group as listed in Scheme 1 and the pharmacologically active salts thereof.
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申请公布号 |
CA2417904(A1) |
申请公布日期 |
2002.02.14 |
申请号 |
CA20012417904 |
申请日期 |
2001.08.07 |
申请人 |
MELACURE THERAPEUTICS AB |
发明人 |
KALVINS, IVARS;BOMAN, ARNE;SKOTTNER, ANNA;LUNDSTEDT, TORBJORN;ANDRIANOV, VICTOR;ANDERSSON, PER |
分类号 |
A61K31/155;A61K31/40;A61K31/4045;A61K31/44;A61K31/4439;A61K45/00;A61P3/04;A61P3/10;A61P5/00;A61P7/00;A61P15/00;A61P25/00;A61P25/18;A61P29/00;A61P37/08;C07C281/18;C07D207/335;C07D209/14;C07D209/40;C07D213/53;C07D213/74;C07D401/12;C07D405/12;(IPC1-7):C07C281/18;C07D213/36 |
主分类号 |
A61K31/155 |
代理机构 |
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代理人 |
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地址 |
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