| 发明名称 |
NOVEL HETEROCYCLIC COMPOUNDS AND THEIR USE AS MEDICINES |
| 摘要 |
The invention concerns novel heterocyclic derivatives having a calpain inhibiting activity and/or an activity trapping reactive oxygen species, of formula (I) wherein A, X, Y, R<1>, R<2> and Het represent variable groups. The invention also concerns methods for preparing said compounds, pharmaceutical preparations containing them and their therapeutic use, in particular as calpain inhibitors and/or as trapping agents for reactive oxygen species, whether selectively or not.
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| 申请公布号 |
WO0132654(A3) |
申请公布日期 |
2001.09.27 |
| 申请号 |
WO2000FR03067 |
申请日期 |
2000.11.03 |
| 申请人 |
SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.);AUVIN, SERGE;CHABRIER DE LASSAUNIERE, PIERRE-ETIENNE |
发明人 |
AUVIN, SERGE;CHABRIER DE LASSAUNIERE, PIERRE-ETIENNE |
| 分类号 |
C07D317/46;A61K31/34;A61K31/341;A61K31/343;A61K31/35;A61K31/353;A61K31/40;A61K31/4025;A61K31/404;A61K31/42;A61K31/421;A61K31/422;A61K31/536;A61K31/5415;A61P3/10;A61P9/00;A61P9/08;A61P9/10;A61P19/10;A61P21/00;A61P25/00;A61P25/02;A61P27/12;A61P29/00;A61P31/12;A61P31/18;A61P37/00;A61P37/02;A61P39/06;C07D;C07D263/18;C07D263/24;C07D307/22;C07D307/24;C07D405/12;C07D407/12;C07D409/12;C07D413/12;C07D417/12;C07D417/14;(IPC1-7):C07D407/12 |
主分类号 |
C07D317/46 |
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