发明名称 |
METAL-CATALYZED ARYLATIONS AND VINYLATIONS OF HYDRAZINES, HYDRAZONES, HYDROXYLAMINES AND OXIMES |
摘要 |
A method is provided for the transition metal-catalyzed arylation, or vinylation, of hydrazines, hydrazones, and the like. Additionally, the invention provides a conceptually novel strategy, the cornerstone of which is the transition metal-catalyzed arylation or vinylation method, for the synthesis of indoles, carbazoles, and the like. The methods and strategies of the invention may be utilized in standard, parallel, and combinatorial synthetic protocols. |
申请公布号 |
EP1058678(A2) |
申请公布日期 |
2000.12.13 |
申请号 |
EP19990908515 |
申请日期 |
1999.02.26 |
申请人 |
MASSACHUSETTS INSTITUTE OF TECHNOLOGY |
发明人 |
BUCHWALD, STEPHEN L.;WAGAW, SEBLE;GEIS, OLIVER |
分类号 |
C07D307/36;C07B61/00;C07C241/02;C07C241/04;C07C243/00;C07C243/22;C07C243/28;C07C249/16;C07C251/84;C07C251/86;C07C255/66;C07C281/08;C07D207/323;C07D209/08;C07D209/60;C07D209/86;C07D213/77;C07D307/79;C07D401/04;(IPC1-7):C07C243/00 |
主分类号 |
C07D307/36 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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