发明名称 |
PARTICLE-FORMING COMPOSITIONS CONTAINING FUSED PYRROLOCARBAZOLES |
摘要 |
A non-aqueous, particle-forming, fused pyrrolocarbazole-containing composition is disclosed. Upon contact with an aqueous medium, the particle-forming composition spontaneously disperses into suspended particles, thereby forming a stable suspension that provides greatly improved bioavailability of orally administered fused pyrrolocarbazole compounds. |
申请公布号 |
WO0008004(A8) |
申请公布日期 |
2000.06.22 |
申请号 |
WO1999US17795 |
申请日期 |
1999.08.06 |
申请人 |
CEPHALON, INC. |
发明人 |
DICKASON, DAVID, A.;PATEL, PIYUSH, R.;CORVARI, VINCENT;SHEK, EFRAIM;HERMAN, JOSEPH, L.;SKELL, JEFFRY, M. |
分类号 |
A61K9/10;A61K31/40;A61K31/403;A61K31/55;A61K31/5513;A61K31/553;A61K47/10;A61K47/12;A61K47/14;A61K47/34;A61K47/44;A61P25/00;A61P35/00;C07D273/06;C09B5/00 |
主分类号 |
A61K9/10 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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