| 摘要 |
<p>(A) alpha-(Aminoalkoxyphenyl)-alpha'-nitrostilbenes of formula: (I) A = ethylene or propylene; R1 and R2 singly = alkyl; or R1 and R2 together = oxydiethylene or alkylene (C4-C8) of which 4 or 5 C atoms form a ring with the N-atom; R3 and R4 = H, halogen, alkyl, alkoxy, CF3. (B) Acid addn. salts of (I). (C) Quaternary ammonium salts of (I). Anti-oestrogenic and hypocholesterolaemic agents for oral or parenteral admin. Prefd. anti-oestrogen is alpha-(p-(2-pyrrolidinoethoxy)-phenyl)-alpha'-nitro-4-methoxy stilbene, prefd. hypocholesterolaemic is alpha-p-(2-diethylaminoethoxy)-phenyl)-alpha'-nitro-4-methoxy-sti- lbene.</p> |
