发明名称 |
Phospholipid deriv. with drug attached at 2 position |
摘要 |
Phospholipid analogues of formula (I) and their water-soluble salts are new. X = H, CH2CH2NH2, CH2CH2N<+>Me3 or CH2CH(NH2)COOH; Y = pharmaceutically active cpd. attached via a carbonyl gp. or via a bridging element (BE). Also new are (1) a BE-contg. active ingredient or steroid prodrug of formula (II) as starting materials for (I). Z = Me or CH2Ph; W = CO(CH2)nCOOH; n is not defined.
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申请公布号 |
CH685284(A5) |
申请公布日期 |
1995.05.31 |
申请号 |
CH19900003690 |
申请日期 |
1990.11.21 |
申请人 |
DR. TUERKAN ELDEM C/O DR. NUR OEZMELPROF. DR. PETER PAUL SPEISER EK |
发明人 |
ELDEM, TUERKAN, DR.;SPEISER, PETER PAUL, PROF. DR. |
分类号 |
C07F9/10;C07J1/00;C07J51/00;(IPC1-7):A61K31/66;A61K47/24;C07F9/09 |
主分类号 |
C07F9/10 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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