发明名称 Phospholipid deriv. with drug attached at 2 position
摘要 Phospholipid analogues of formula (I) and their water-soluble salts are new. X = H, CH2CH2NH2, CH2CH2N<+>Me3 or CH2CH(NH2)COOH; Y = pharmaceutically active cpd. attached via a carbonyl gp. or via a bridging element (BE). Also new are (1) a BE-contg. active ingredient or steroid prodrug of formula (II) as starting materials for (I). Z = Me or CH2Ph; W = CO(CH2)nCOOH; n is not defined.
申请公布号 CH685284(A5) 申请公布日期 1995.05.31
申请号 CH19900003690 申请日期 1990.11.21
申请人 DR. TUERKAN ELDEM C/O DR. NUR OEZMELPROF. DR. PETER PAUL SPEISER EK 发明人 ELDEM, TUERKAN, DR.;SPEISER, PETER PAUL, PROF. DR.
分类号 C07F9/10;C07J1/00;C07J51/00;(IPC1-7):A61K31/66;A61K47/24;C07F9/09 主分类号 C07F9/10
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