发明名称 |
TAXANES HAVING ALKOXY, ALKENOXY OR ARYLOXY SUBSTITUTED SIDE-CHAIN AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME |
摘要 |
<p>Taxane derivatives having a C13 side chain which includes an N-substituted group and the formula of the group is -COOX10 wherein X10 is alkyl, alkenyl or aryl. The taxane derivatives are useful antileukemia and anticancer agents.</p> |
申请公布号 |
WO9421250(A1) |
申请公布日期 |
1994.09.29 |
申请号 |
WO1994US03053 |
申请日期 |
1994.03.21 |
申请人 |
FLORIDA STATE UNIVERSITY |
发明人 |
HOLTON, ROBERT, A.;NADIZADEH, HOSSAIN;CHAI, KI-BYUNG;RENGAN, KASTHURI;SUZUKI, YUKIO;TAO, CHUNLIN;IDMOUMAZ, HAMID |
分类号 |
C07D333/20;A61K31/335;A61K31/337;A61K31/34;A61K31/341;A61K31/38;A61K31/381;A61P35/00;A61P35/02;C07C227/22;C07C231/12;C07C233/87;C07D205/08;C07D205/085;C07D205/09;C07D305/14;C07D307/00;C07D401/04;C07D401/12;C07D401/14;C07D403/04;C07D403/12;C07D403/14;C07D405/04;C07D405/12;C07D405/14;C07D407/00;C07D407/12;C07D407/14;C07D409/00;C07D409/04;C07D409/12;C07D409/14;C07D413/14;C07F7/08;C07F7/18;(IPC1-7):A61K31/335 |
主分类号 |
C07D333/20 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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