发明名称 NOVEL MERCAPTOACETYLAMIDO PYRIDAZO[1,2]PYRIDAZINE, PYRAZOLO[1,2]PYRIDAZINE, PYRIDAZO[1,2-a][1,2]DIAZEPINE AND PYRAZOLO[1,2-a][1,2]DIAZEPINE DERIVATIVES USEFUL AS INHIBITORS OF ENKEPHALINASE AND ACE
摘要 The present invention relates to certain novel mercaptoacetylamido pyridazo[1,2]pyridazine, pyrazolo[1,2]pyridazine, pyridazo[1,2-a][1,2]diazepine and pyrazolo[1,2-a][1,2]diazepine derivatives of formula (I) useful as inhibitors of enkephalinase and of ACE.
申请公布号 WO9323403(A1) 申请公布日期 1993.11.25
申请号 WO1993US03721 申请日期 1993.04.21
申请人 MERRELL DOW PHARMACEUTICALS INC. 发明人 FLYNN, GARY, A.;SHUM, PATRICK, W.
分类号 A61K31/415;A61K31/50;A61K31/5025;A61K31/55;A61K38/00;A61P7/10;A61P9/00;A61P9/12;A61P25/04;A61P25/24;A61P25/28;A61P43/00;C07D487/04;C07K5/078;(IPC1-7):C07D487/04 主分类号 A61K31/415
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