发明名称 FOERFARANDE FOER FRAMSTAELLNING AV NYA TERAPEUTISKT ANVAENDBARA 1,2-BENZISOTIAZOL-3-YLPIPERAZINDERIVAT.
摘要 A series of non-opiate analgesics of Formula I <IMAGE> I wherein R1 is hydrogen, alkyl, aralkyl, or aryloxyalkyl; R2 is alkyl or hydrogen; and R3 and R4 are independently selected from hydrogen, alkyl, acyloxy, alkoxy, alkylthio, halogen, hydroxyl, or trifluoromethyl; or a pharmaceutically acceptable acid addition salt.
申请公布号 FI82039(B) 申请公布日期 1990.09.28
申请号 FI19850003193 申请日期 1985.08.20
申请人 SQUIBB BRISTOL-MYERS CO 发明人 SMITH DAVID W;YEVICH JOSEPH P
分类号 A61K31/425;A61K31/428;A61K31/495;A61P25/02;A61P25/04;A61P25/20;C07D275/04;C07D319/00;C07D417/04;C07D417/12 主分类号 A61K31/425
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