发明名称 Tetrazole deriv. prepn.
摘要 1H-Tetrazole cpds. of formula (I), in which A is carbonyl or 2-4C methylene, P is a pyridine ring, X1 and X2 are halogen, 1-4C alkyl or other, and Y is O, S or other, are made by reacting a cpd. of formula (II) with hydrazoic acid in DMF in presence of BCl3 etherate at 10-200 deg.C for 5-24 hours, to obtain (I) or its acceptable salts.
申请公布号 ES8707229(A3) 申请公布日期 1987.10.01
申请号 ES19790005564 申请日期 1986.06.23
申请人 YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. 发明人
分类号 A61K31/35;A61K31/41;A61K31/44;C07D405/14;(IPC1-7):C07D405/14 主分类号 A61K31/35
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