发明名称 PYRIMIDINE COMPOUND CRYSTAL OR AMORPHOUS FORM AND PROCESS FOR PRODUCING THE SAME
摘要 Crystal of 5-[2-amino-4-(2-furyl)pyrimidin-5-yl]-1-methylpyridin-2(1H)-one exhibiting, in powder X-ray diffractometry, diffraction peaks at diffraction angles (2theta±0.2°) of 9.7° and/or 21.9°. This crystal is suitable for use as an active ingredient of preventive/therapeutic agents for diseases, such as costiveness. Further, a hydrate of 5-[2-amino-4-(2-furyl)pyrimidin-5-yl]-1-methylpyridin-2(1H)-one and 5-[2-amino-4-(2-furyl) pyrimidin-5-yl]-1-methylpyridin-2(1H)-one in amorphous form are also suitable for use as an active ingredient of preventive/therapeutic agents for diseases, such as costiveness.
申请公布号 KR20070112368(A) 申请公布日期 2007.11.23
申请号 KR20077016421 申请日期 2007.07.18
申请人 EISAI R&D MANAGEMENT CO., LTD. 发明人 HARADA HITOSHI;ISHIHARA HIROSHI;SATO YOSHIAKI;CHIBA HIROYUKI;KOMATSU YUKI;INOUE SUSUMU;OZEKI NAOKI
分类号 C07D405/14 主分类号 C07D405/14
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