发明名称 TRYPSIN-LIKE SERINE PROTEASE INHIBITORS, AND THEIR PREPARATION AND USE
摘要 The invention relates to inhibitors of trypsin-like serine proteases of the general formula (I) which, as well as plasmin, also inhibit plasma kallikrien, and to their preparation and use as medicaments, preferably for treatment of blood loss, especially in the case of hyperfibrinolytic states, in organ transplants or heart surgery interventions, in particular with a cardiopulmonary bypass, or as a constituent of a fibrin adhesive.
申请公布号 US2010022781(A1) 申请公布日期 2010.01.28
申请号 US20090429766 申请日期 2009.04.24
申请人 STEINMETZER TORSTEN;SCHWEINITZ ANDREA;STUERZEBECHER JOERG;STEINMETZER PETER;SOFFING ANETT;VAN DE LOCHT ANDREAS;NICKLISCH SILKE;REICHELT CLAUDIA;LUDWIG FRIEDRICH-ALEXANDER;SCHULZE ALEXANDER;DAGHISCH MOHAMMED;HEINICKE JOCHEN 发明人 STEINMETZER TORSTEN;SCHWEINITZ ANDREA;STUERZEBECHER JOERG;STEINMETZER PETER;SOFFING ANETT;VAN DE LOCHT ANDREAS;NICKLISCH SILKE;REICHELT CLAUDIA;LUDWIG FRIEDRICH-ALEXANDER;SCHULZE ALEXANDER;DAGHISCH MOHAMMED;HEINICKE JOCHEN
分类号 C07C311/13;C07D233/64 主分类号 C07C311/13
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