摘要 |
<p>(1) Processes detailed below for prepn. of benzodiazepin-2-ones (I) and benzoxadiazocines (II) A = R2-phenyl, lower alkyl, cycloalkyl C3-C7, R, R1, R2 = H, halogen, NO2, CF3, lower alkyl R3, R4 = H, lower alkyl (2) Novels cpds. (II) (3) Novel intermediates (III) and (IV) R' = H, lower alkyl Cpds. (I) are therapeutic agents. Cpds. (II) are anticonvulsants, sedatives, muscle relaxants, and intermediates for cpds. (I).</p> |