发明名称 GEMINALLY SUBSTITUTED CYANOETHYLPYRAZOLO PYRIDONES AS JANUS KINASE INHIBITORS
摘要 The instant invention provides compounds of Formula (I) which are JAK inhibitors, and as such are useful for the treatment of JAK-mediated diseases such as rheumatoid arthritis, asthma, COPD and cancer.
申请公布号 WO2014146491(A1) 申请公布日期 2014.09.25
申请号 WO2014CN00297 申请日期 2014.03.19
申请人 MERCK SHARP & DOHME CORP.;CHILDERS, MATTHEW LLOYD;FULLER, PETER;GUERIN, DAVID;KATZ, JASON DAVID;PU, QINGLIN;SCOTT, MARK E.;THOMPSON, CHRISTOPHER F.;MARTINEZ, MICHELLE;FALCONE, DANIELLE;TORRES, LUIS;DENG, YONGQI;KURUKLASURIYA, RAVI;ZENG, HONGBO;BAI, YUNFENG;KONG, NORMAN;LIU, YUMEI;ZHENG, ZHIXIANG 发明人 CHILDERS, MATTHEW LLOYD;FULLER, PETER;GUERIN, DAVID;KATZ, JASON DAVID;PU, QINGLIN;SCOTT, MARK E.;THOMPSON, CHRISTOPHER F.;MARTINEZ, MICHELLE;FALCONE, DANIELLE;TORRES, LUIS;DENG, YONGQI;KURUKLASURIYA, RAVI;ZENG, HONGBO;BAI, YUNFENG;KONG, NORMAN;LIU, YUMEI;ZHENG, ZHIXIANG
分类号 C07D471/04;A61K31/437;A61K31/444;A61P19/02;A61P29/00;A61P37/00;C07D205/04;C07D211/00;C07D309/02 主分类号 C07D471/04
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