发明名称 |
NONHYGROSCOPIC LINEZOLID SALTS |
摘要 |
<p>The present invention relates to an acid addition salt of linezolid with naphthalene- 1,5-disulfonic acid or with p-toluene sulfonic acid such as linezolid mono-naphtalene-1,5- disulfonate (linezolid hydrogennapadisylate), linezolid hemi-naphthalene-l,5-disulfonate (linezolide napadisylate) and linezolid p-toluene sulfonate (linezolid tosylate), to pharmaceutical compositions comprising them, to a process for making them, to a process for making linezolid base, to the use in making a medicine and use in medicine.</p> |
申请公布号 |
WO2011029460(A1) |
申请公布日期 |
2011.03.17 |
申请号 |
WO2009EP06587 |
申请日期 |
2009.09.09 |
申请人 |
SYNTHON B.V.;WESTHEIM, RAYMOND, JOZEF, HUBERTUS |
发明人 |
WESTHEIM, RAYMOND, JOZEF, HUBERTUS |
分类号 |
C07D263/20;A61K31/5375;A61P31/04 |
主分类号 |
C07D263/20 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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