发明名称 NONHYGROSCOPIC LINEZOLID SALTS
摘要 <p>The present invention relates to an acid addition salt of linezolid with naphthalene- 1,5-disulfonic acid or with p-toluene sulfonic acid such as linezolid mono-naphtalene-1,5- disulfonate (linezolid hydrogennapadisylate), linezolid hemi-naphthalene-l,5-disulfonate (linezolide napadisylate) and linezolid p-toluene sulfonate (linezolid tosylate), to pharmaceutical compositions comprising them, to a process for making them, to a process for making linezolid base, to the use in making a medicine and use in medicine.</p>
申请公布号 WO2011029460(A1) 申请公布日期 2011.03.17
申请号 WO2009EP06587 申请日期 2009.09.09
申请人 SYNTHON B.V.;WESTHEIM, RAYMOND, JOZEF, HUBERTUS 发明人 WESTHEIM, RAYMOND, JOZEF, HUBERTUS
分类号 C07D263/20;A61K31/5375;A61P31/04 主分类号 C07D263/20
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