发明名称 NOVEL PROCESS FOR PREPARING PURE 6-FLUORO-3-PIPERIDIN-4-YL-1,2-BENZISOXAZOLE HYDROCHLORIDE AND ITS CONVERSION TO PALIPERIDONE
摘要 The invention relates to novel process for providing substantially pure 6-Fluoro-3- piperidin-4-yl-1,2-benzisoxazole hydrochloride and its conversion to Paliperidone having dimer compound of structural formula-1 A is less than 0.2 % and HPLC purity > 99.7%.
申请公布号 WO2010082110(A3) 申请公布日期 2010.09.10
申请号 WO2010IB00041 申请日期 2010.01.12
申请人 CADILA PHARMACEUTICALS LTD;SODAGAR, KEVAL, RAMESHCHANDRA;MALIK, VINEET;KAPADIA, BRIJESH NITINKUMAR;JAIN, SUDHIR HUKAMCHAND;PARIKH, SANJAY NATVARLAL;SHARMA, ARUN OMPRAKASH;BAPAT, UDAY RAJARAM;KHAMAR, BAKULESH MAFATIAL 发明人 SODAGAR, KEVAL, RAMESHCHANDRA;MALIK, VINEET;KAPADIA, BRIJESH NITINKUMAR;JAIN, SUDHIR HUKAMCHAND;PARIKH, SANJAY NATVARLAL;SHARMA, ARUN OMPRAKASH;BAPAT, UDAY RAJARAM;KHAMAR, BAKULESH MAFATIAL
分类号 A01N43/90 主分类号 A01N43/90
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