发明名称 |
BICYCLO-PYRAZOLE AS KINASE INHIBITOR, METHOD FOR PRODUCING THE SAME AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME |
摘要 |
PROBLEM TO BE SOLVED: To provide a novel compound useful for treating diseases associated with dysregulated protein kinases. SOLUTION: A bicyclo-pyrazole expressed by formula (I) and having kinase inhibition activity, a pharmaceutically accepted salt of the same and a pharmaceutical composition comprising the same are provided. COPYRIGHT: (C)2010,JPO&INPIT
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申请公布号 |
JP2010111677(A) |
申请公布日期 |
2010.05.20 |
申请号 |
JP20090287171 |
申请日期 |
2009.12.18 |
申请人 |
PFIZER ITALIA SRL |
发明人 |
FANCELLI DANIELE;PITTALA VALERIA;VARASI MARIO |
分类号 |
C07D471/04;A61K31/4162;A61K31/4178;A61K31/4192;A61K31/423;A61K31/427;A61K31/437;A61K31/4439;A61K31/454;A61K31/4545;A61K31/4709;A61K31/496;A61K31/497;A61K31/498;A61K31/501;A61K31/5377;A61P9/00;A61P9/10;A61P11/00;A61P13/08;A61P13/12;A61P17/06;A61P19/02;A61P25/00;A61P25/28;A61P29/00;A61P31/12;A61P35/00;A61P35/02;A61P35/04;A61P37/02;A61P43/00;C07B61/00;C07D487/04;C40B40/04 |
主分类号 |
C07D471/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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