发明名称 NOVEL MCH RECEPTOR ANTAGONISTS
摘要 The present invention relates to a melanin concentrating hormone antagonist compound of formula (I): wherein R1, Ra, Rb, R2, L1, R3, R4 and R5 are as defined, or a pharmaceutically acceptable salt, enantiomer, diastereomer or mixture of diastereomers thereof useful in the treatment, obesity and related diseases.
申请公布号 US2010016350(A1) 申请公布日期 2010.01.21
申请号 US20070296557 申请日期 2007.06.08
申请人 AMEGADZIE ALBERT KUDZOVI;DAO YEN;GARDINIER KEVIN MATTHEW;GARMENE DAVID JOSEPH;GREEN STEVEN JAMES;HEMBRE ERIK JAMES;LU JIANLAING;SPINAZZE PATRICK GIANPIETRO 发明人 AMEGADZIE ALBERT KUDZOVI;DAO YEN;GARDINIER KEVIN MATTHEW;GARMENE DAVID JOSEPH;GREEN STEVEN JAMES;HEMBRE ERIK JAMES;LU JIANLAING;SPINAZZE PATRICK GIANPIETRO
分类号 A61K31/4365;A61P3/04;C07D495/04 主分类号 A61K31/4365
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