发明名称 3,2-benzoxazepines
摘要 Title cpds. formula (I) (where R is H or 1-4C alkyl, R1 is H, 1-4C alkyl opt. substd. by OH, 3-5C alkenyl, opt. substd. carbamoy-: loxyalkyl, acyl, amidino or opt. substd. carbamoyl, and R2 is H, NO2, NH2 acylamino or halogen in the 7- or 8-posn) are prepd. by cyclisation of a cpd. (II) (where R3 is alkyl or aralkyl) in the presence of a base and opt. hydrolysis (I; R1 = COOR3) or by nitrating (I; R2 = H) reducing nitro to amino and acylating amino or replacing by halogen.
申请公布号 CH536852(A) 申请公布日期 1973.05.15
申请号 CH19730003645 申请日期 1972.03.16
申请人 GRUPPO LEPETIT S. P. A. 发明人 PIFFERI,GIORGIO;OMODEI-SALE,AMADEO;CONSONNI,PIETRO
分类号 C07D267/04;C07D267/14;(IPC1-7):C07D87/54 主分类号 C07D267/04
代理机构 代理人
主权项
地址