发明名称 QUINOXALINE AND QUINOLINE DERIVATIVES AS KINASE INHIBITORS
摘要 <p>A series of heteroaryl-substituted quinoxaline and quinoline derivatives, being selective inhibitors of PI3 kinase enzymes, are accordingly of benefit in medicine, for example in the treatment of inflammatory, autoimmune, cardiovascular, neurodegenerative, metabolic, oncological, nociceptive or ophthalmic conditions.</p>
申请公布号 WO2009081105(A3) 申请公布日期 2009.08.20
申请号 WO2008GB04171 申请日期 2008.12.17
申请人 UCB PHARMA S.A.;ALLEN, DANIEL, REES;BUCKLEY, GEORGE, MARTIN;BUERLI, ROLAND;DAVENPORT, RICHARD, JOHN;KINSELLA, NATASHA;LOCK, CHRISTOPHER, JAMES;LOWE, CHRISTOPHER;MACK, STEPHEN, ROBERT;PITT, WILLIAM, ROSS;RATCLIFFE, ANDREW, JAMES;RICHARD, MARIANNA, DILANI;SABIN, VERITY, MARGARET;SHARPE, ANDREW;TAIT, LAURA, JANE;WARRELOW, GRAHAM, JOHN;WILLIAMS, SOPHIE, CAROLINE 发明人 ALLEN, DANIEL, REES;BUCKLEY, GEORGE, MARTIN;BUERLI, ROLAND;DAVENPORT, RICHARD, JOHN;KINSELLA, NATASHA;LOCK, CHRISTOPHER, JAMES;LOWE, CHRISTOPHER;MACK, STEPHEN, ROBERT;PITT, WILLIAM, ROSS;RATCLIFFE, ANDREW, JAMES;RICHARD, MARIANNA, DILANI;SABIN, VERITY, MARGARET;SHARPE, ANDREW;TAIT, LAURA, JANE;WARRELOW, GRAHAM, JOHN;WILLIAMS, SOPHIE, CAROLINE
分类号 C07D401/14;A61K31/395;A61P35/00;C07D403/06;C07D403/12;C07D403/14;C07D409/14;C07D413/14;C07D473/34;C07D473/36 主分类号 C07D401/14
代理机构 代理人
主权项
地址