发明名称 METABOLITES OF 5-FLUORO-8-{4-[4-(6-METHOXYQUINOLIN-8-YL)PIPERAZIN-1-YL]PIPERIDIN-1-YL} QUINOLINE AND METHODS OF PREPARATION AND USES THEREOF
摘要 The present invention relates to novel metabolites of 5-Fluoro-8-{4-[4-(6- methoxyquinolin-8-yl)piperazin-l-yl]piperidin-l -yl}quinoline, which can be useful in treating CNS disorders. The present invention further relates to processes for their preparation, to pharmaceutical compositions comprising them, and to methods of using them.
申请公布号 WO2008067390(A9) 申请公布日期 2009.05.22
申请号 WO2007US85777 申请日期 2007.11.28
申请人 WYETH;WANG, JIANYAO;UPTHAGROVE, ALANA;DENG, LIN;CHILDERS, WAYNE, EVERETT;SHEN, ZHONGQI;DEMAIO, WILLIAM;MOORE, ROBIN, D.;TONG, ZEEN;SHEN, LI;LI, PIXU;MAY, MICHAEL, K. 发明人 WANG, JIANYAO;UPTHAGROVE, ALANA;DENG, LIN;CHILDERS, WAYNE, EVERETT;SHEN, ZHONGQI;DEMAIO, WILLIAM;MOORE, ROBIN, D.;TONG, ZEEN;SHEN, LI;LI, PIXU;MAY, MICHAEL, K.
分类号 C07D401/12;A61K31/4709;A61P25/00;C07D405/14 主分类号 C07D401/12
代理机构 代理人
主权项
地址