发明名称 |
Novel crystals and process of making 5-({[2-amino-3-(4-carbamoyl-2,6-dimethyl-phenyl)-propionyl]-[1-(4-phenyl-1h-imidazol-2-yl)-ethyl]-amino}-methyl)-2-methoxy- benzoic acid |
摘要 |
<p>The present invention relates to a novel crystals of 5-({[2-amino-3-(4-carbamoyl-2,6-dimethyl-phenyl)-propionyl]-[1-(4-phenyl-1h-imidazol-2-yl)-ethyl]-amino}-methyl)-2-methoxy-benzoic acid and methods of making the zwitterion of 5-({[2-amino-3-(4-carbamoyl-2,6-dimethyl-phenyl)-propionyl]-[1-(4-phenyl-1h-imidazol-2-yl)-ethyl]-amino}-methyl)-2-methoxy-benzoic acid.</p> |
申请公布号 |
AU2008275270(A1) |
申请公布日期 |
2009.01.15 |
申请号 |
AU20080275270 |
申请日期 |
2008.07.07 |
申请人 |
JANSSEN PHARMACEUTICA N.V. |
发明人 |
CHRISTOPHER ALLAN TELEHA;FRANK J. VILLANI;LUIGI ANZALONE;PENINA FEIBUSH;BARRY FEGELY |
分类号 |
A61K31/4164;A61P1/00;C07D233/64 |
主分类号 |
A61K31/4164 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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