发明名称 |
Benzamide derivatives as oxytocin agonists and vasopressin antagonists |
摘要 |
Novel compounds according to general formula 1, wherein G<SUP>1 </SUP>is NR<SUP>5</SUP>R<SUP>6 </SUP>or a fused polycyclic group that are specific OT receptor agonists and/or V<SUB>1a </SUB>receptor antagonists. Pharmaceutical compositions comprising such compounds are useful in the treatment of, inter alia, primary dysmenorrhoea.
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申请公布号 |
US2008275026(A1) |
申请公布日期 |
2008.11.06 |
申请号 |
US20080213576 |
申请日期 |
2008.06.20 |
申请人 |
FERRING B.V. |
发明人 |
HUDSON PETER;BATT ANDRZEJ ROMAN;HEENEY CELINE MARGUERITE SIMONE;BAXTER ANDREW JOHN;ROE MICHAEL BRYAN;ROBSON PETER ANDREW |
分类号 |
A61K31/5513;A61K31/55;A61K31/5517;A61P15/00;C07D223/14;C07D471/04;C07D471/14;C07D487/04;C07D487/14;C07D495/04;C07D498/04 |
主分类号 |
A61K31/5513 |
代理机构 |
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地址 |
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