发明名称 Benzamide derivatives as oxytocin agonists and vasopressin antagonists
摘要 Novel compounds according to general formula 1, wherein G<SUP>1 </SUP>is NR<SUP>5</SUP>R<SUP>6 </SUP>or a fused polycyclic group that are specific OT receptor agonists and/or V<SUB>1a </SUB>receptor antagonists. Pharmaceutical compositions comprising such compounds are useful in the treatment of, inter alia, primary dysmenorrhoea.
申请公布号 US2008275026(A1) 申请公布日期 2008.11.06
申请号 US20080213576 申请日期 2008.06.20
申请人 FERRING B.V. 发明人 HUDSON PETER;BATT ANDRZEJ ROMAN;HEENEY CELINE MARGUERITE SIMONE;BAXTER ANDREW JOHN;ROE MICHAEL BRYAN;ROBSON PETER ANDREW
分类号 A61K31/5513;A61K31/55;A61K31/5517;A61P15/00;C07D223/14;C07D471/04;C07D471/14;C07D487/04;C07D487/14;C07D495/04;C07D498/04 主分类号 A61K31/5513
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