发明名称 BENZIMIDAZOLE-CARBOXAMIDE COMPOUNDS AS 5-HT4 RECEPTOR AGONISTS.
摘要 The invention relates to benzimidazole-carboxamide 5-HT<sub>4</sub> receptor agonist compounds of formula (I), wherein R<sup>1</sup> and X are as defined in the specification, or a pharmaceutically acceptable salt or solvate or stereoisomer thereof. The invention also relates to pharmaceutical compositions comprising such compounds, methods of using such compounds to treat diseases associated with 5-HT<sub>4</sub> receptor activity, and processes and intermediates useful for preparing such compounds. The invention further relates to crystalline forms of a compound of formula (I).
申请公布号 MX2007014762(A) 申请公布日期 2008.02.14
申请号 MX20070014762 申请日期 2006.05.24
申请人 THERAVANCE, INC. 发明人 ROBERT MURRAY MCKINNELL.;DANIEL D. LONG.;DANIEL MARQUESS;SEOK-KI CHOI;PAUL R. FATHEREE;ROLAND GENDRON;LAN JIANG;SEAN M. DALZIEL;KIRSTEN M. PHIZACKERLEY
分类号 C07D401/14;A61K31/4545;A61P1/00;C07D405/14;C07D409/14 主分类号 C07D401/14
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