发明名称 A PROCESS FOR THE PREPARATION OF TETRAZOLYLTETRAHYDROCYCLOPENTAPYRAZOLES
摘要 <p>A process for the preparation of a compound of formula (I), or a salt, hydrate or solvate thereof; wherein R&lt;SUP&gt;1&lt;/SUP&gt; and R&lt;SUP&gt;2 &lt;/SUP&gt;are each independently hydrogen, or C&lt;SUB&gt;1-6 &lt;/SUB&gt;alkyl groups or R&lt;SUP&gt;1&lt;/SUP&gt; and R&lt;SUP&gt;2&lt;/SUP&gt; are linked and, together with the cyclopentane carbon atoms to which they are attached, form a cyclopropyl ring.</p>
申请公布号 WO2006114581(A1) 申请公布日期 2006.11.02
申请号 WO2006GB01446 申请日期 2006.04.20
申请人 MERCK SHARP & DOHME LIMITED;ASHWOOD, MICHAEL, STEWART;BIO, MATTHEW;CLEATOR, EDWARD;HANDS, DAVID;SHEEN, FAYE, JULIA;WILSON, ROBERT, DARRIN 发明人 ASHWOOD, MICHAEL, STEWART;BIO, MATTHEW;CLEATOR, EDWARD;HANDS, DAVID;SHEEN, FAYE, JULIA;WILSON, ROBERT, DARRIN
分类号 C07D403/04 主分类号 C07D403/04
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