发明名称 |
One-pot synthesis of alkyl 3-cyclopropylamino-2-Ä2,4-dibromo-3-(difluoromethoxy)benzoylÜ-2-propenoate as a useful intermediate for antibacterial quinolone medicaments |
摘要 |
The present invention relates to a new and industrially advantageous one-pot process for the preparation of alkyl 3-cyclopropyl amino-2-[2,4-dibromo-3-(difluoromethoxy) benzoyl]-2-propenoates in which R represents methyl or ethyl, which are valuable intermediates for the production of highly active antibacterial quinolone medicaments. |
申请公布号 |
US6835848(B1) |
申请公布日期 |
2004.12.28 |
申请号 |
US20030221113D |
申请日期 |
2003.01.06 |
申请人 |
RANBAXY LABORATORIES LIMITED;TOYAMA CHEMICAL CO., LTD. |
发明人 |
BOSE PROSENJIT;KUMAR NARESH;KIYOTO TARO |
分类号 |
C07C227/18;C07C227/16;C07C229/34;(IPC1-7):C07C229/00;C07C59/56;C07C65/32 |
主分类号 |
C07C227/18 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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