发明名称 |
THIENOPYRIMIDINES, PROCESS FOR PREPARING THE SAME AND USE THEREOF |
摘要 |
The present invention provides a thienopyrimidine compound, represented by the formula <CHEM> Äwherein, R<1> is C1-4 alkyl, R<2> is (1) phenyl optionally having a substituent such as amino, mono C1-4 alkylamino and di C1-4 alkylamino, or (2) a heterocyclic group optionally having a substituent such as amino, mono C1-4 alkylamino and di C1-4 alkylamino and the like, R<3> is a hydrogen atom or C1-4 alkyl, R<4> is C1-4 alkyl optionally having a substituent such as C1-4 alkoxy-carbonyl, carboxyl, mono C1-4 alkylamino and N-C1-4 alkyl-N-C7-10 aralkylamino and the likeÜ or a salt thereof, which has antagonistic action for gonadotropin-releasing hormone. |
申请公布号 |
EP1479684(A1) |
申请公布日期 |
2004.11.24 |
申请号 |
EP20030734872 |
申请日期 |
2003.01.29 |
申请人 |
TAKEDA CHEMICAL INDUSTRIES, LTD. |
发明人 |
FURUYA, SHUICHI;IMADA, TAKASHI;HITAKA, TAKENORI;MIWA, KAZUHIRO;KUSAKA, MASAMI;SUZUKI, NOBUHIRO |
分类号 |
A61P5/08;A61P5/24;A61P13/08;A61P15/00;A61P15/08;A61P17/10;A61P17/14;A61P25/28;A61P35/00;A61P35/04;A61P43/00;C07D495/04 |
主分类号 |
A61P5/08 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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