发明名称 THIENOPYRIMIDINES, PROCESS FOR PREPARING THE SAME AND USE THEREOF
摘要 The present invention provides a thienopyrimidine compound, represented by the formula <CHEM> Äwherein, R<1> is C1-4 alkyl, R<2> is (1) phenyl optionally having a substituent such as amino, mono C1-4 alkylamino and di C1-4 alkylamino, or (2) a heterocyclic group optionally having a substituent such as amino, mono C1-4 alkylamino and di C1-4 alkylamino and the like, R<3> is a hydrogen atom or C1-4 alkyl, R<4> is C1-4 alkyl optionally having a substituent such as C1-4 alkoxy-carbonyl, carboxyl, mono C1-4 alkylamino and N-C1-4 alkyl-N-C7-10 aralkylamino and the likeÜ or a salt thereof, which has antagonistic action for gonadotropin-releasing hormone.
申请公布号 EP1479684(A1) 申请公布日期 2004.11.24
申请号 EP20030734872 申请日期 2003.01.29
申请人 TAKEDA CHEMICAL INDUSTRIES, LTD. 发明人 FURUYA, SHUICHI;IMADA, TAKASHI;HITAKA, TAKENORI;MIWA, KAZUHIRO;KUSAKA, MASAMI;SUZUKI, NOBUHIRO
分类号 A61P5/08;A61P5/24;A61P13/08;A61P15/00;A61P15/08;A61P17/10;A61P17/14;A61P25/28;A61P35/00;A61P35/04;A61P43/00;C07D495/04 主分类号 A61P5/08
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