| 发明名称 |
Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof |
| 摘要 |
Compounds of Formula (IA) and Formula (IB) wherein R<1>, R<2>, R<3>, R<4>, R<5>, and R<6 >are as defined herein for Formula (IA) or Formula (IB), or a tautomer, prodrug, solvate, or salt thereof; pharmaceutical compositions containing such compounds, and methods of modulating the glucocorticoid receptor function and methods of treating disease-states or conditions mediated by the glucocorticoid receptor function or characterized by inflammatory, allergic, or proliferative processes in a patient using these compounds.
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| 申请公布号 |
US2004029932(A1) |
申请公布日期 |
2004.02.12 |
| 申请号 |
US20030394157 |
申请日期 |
2003.03.21 |
| 申请人 |
BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. |
发明人 |
BEKKALI YOUNES;CARDOZO MARIO G.;HARCKEN CHRISTIAN HANKE JUSTUS JOACHIM;KIRRANE THOMAS M.;KUZMICH DANIEL;PROUDFOOT JOHN ROBERT;RAZAVI HOSSEIN;TAKAHASHI HIDENORI;THOMSON DAVID S.;WANG JI;ZINDELL RENEE |
| 分类号 |
C07D333/62;A61K31/065;A61K31/085;A61K31/09;A61K31/10;A61K31/11;A61K31/121;A61K31/15;A61K31/165;A61K31/166;A61K31/192;A61K31/27;A61K31/277;A61K31/343;A61K31/381;A61K31/4402;A61P1/04;A61P1/16;A61P3/04;A61P3/10;A61P5/00;A61P7/00;A61P7/08;A61P9/00;A61P9/04;A61P9/10;A61P9/12;A61P9/14;A61P11/00;A61P11/02;A61P11/04;A61P13/12;A61P17/00;A61P17/02;A61P19/00;A61P19/02;A61P19/08;A61P25/00;A61P25/04;A61P25/28;A61P27/02;A61P27/06;A61P27/14;A61P27/16;A61P29/00;A61P29/02;A61P31/04;A61P35/00;A61P37/06;A61P37/08;A61P43/00;C07C37/50;C07C39/367;C07C39/373;C07C43/23;C07C45/00;C07C45/30;C07C45/44;C07C45/45;C07C45/63;C07C45/67;C07C45/68;C07C45/69;C07C47/575;C07C49/233;C07C49/255;C07C49/577;C07C49/83;C07C49/84;C07C59/56;C07C65/24;C07C235/42;C07C235/46;C07C251/48;C07C255/53;C07C255/54;C07C317/22;C07C323/18;C07D213/30;C07D307/78;(IPC1-7):C07D213/57;A61K31/44;A61K31/40;A61K31/137 |
主分类号 |
C07D333/62 |
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