发明名称 BENZAMIDES AND RELATED INHIBITORS OF FACTOR XA
摘要 Benzamide compounds of the formulae (VI) and (VII), where the variables are as defined in the claims, including their pharmaceutically acceptable isomers, salts, hydrates, solvates and prodrug derivatives having activity against mammalian factor Xa are described. Compositions containing such compounds ar e also described. The compounds and compositions are useful in vitro or in viv o for preventing or treating coagulation disorders.
申请公布号 CA2401778(A1) 申请公布日期 2001.09.07
申请号 CA20012401778 申请日期 2001.02.28
申请人 COR THERAPEUTICS, INC. 发明人 GOLDMAN, ERICK;ZHANG, PENGLIE;HUANG, WENRONG;ZHU, BING-YAN;WANG, LINGYAN;SCARBOROUGH, ROBERT;SONG, YONGHONG;LI, WENHAO;ZUCKETT, JINGMEI
分类号 A61K31/443;A61K31/444;A61P7/02;C07C311/16;C07C311/46;C07C317/40;C07C317/44;C07D213/75;C07D213/81;C07D213/82;C07D217/22;C07D333/38;C07D401/12;C07D409/12;C07D409/14;C07D521/00 主分类号 A61K31/443
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