发明名称 |
SPIROPIPERIDINE DERIVATIVES, PROCESS OF THEIR PREPARATION AND PHARMACEUTICAL COMPOSITION CONTAINING THEREOF |
摘要 |
<p>PCT No. PCT/GB97/01630 Sec. 371 Date Dec. 16, 1998 Sec. 102(e) Date Dec. 16, 1998 PCT Filed Jun. 17, 1997 PCT Pub. No. WO97/49710 PCT Pub. Date Dec. 31, 1997The present invention relates to certain spiro-piperdine derivatives which are tachykinnin antagonists and are useful, for example, in the treatment or prevention of pain, inflammation, migraine, emesis and postherpetic neuralgia.</p> |
申请公布号 |
CZ9804247(A3) |
申请公布日期 |
1999.05.12 |
申请号 |
CZ19980004247 |
申请日期 |
1997.06.17 |
申请人 |
MERCK SHARP AND DOHME LIMITED |
发明人 |
BAKER RAYMOND;CURTIS NEIL ROY;ELLIOTT JASON MATTHEW;HARRISON TIMOTHY;HOLLINGWORTH GREGORY JOHN;JACKSON PHILIP STEPHEN;KULAGOWSKI JANUSZ JOZEF;SEWARD EILEEN MARY;SWAIN CHRISTOPHER JOHN;WILLIAMS BRIAN JOHN |
分类号 |
A61K31/00;A61K31/395;A61K31/435;A61K31/438;A61K31/445;A61K31/451;A61K31/5375;A61K31/5377;A61K31/675;A61P1/00;A61P1/08;A61P25/04;A61P25/06;A61P29/00;A61P43/00;C07D211/56;C07D491/10;C07D491/107;(IPC1-7):C07D491/10 |
主分类号 |
A61K31/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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