发明名称 |
BENZODIAZEPINE DERIVATIVES |
摘要 |
Benzodiazepine derivatives of formula (I) wherein R<1> is aryl which may have one or more suitable substituent(s), R<2> is C3-C8 cycloalkyl which may have one or more suitable substituent(s), A is lower alkylene, R<3> is a heterocyclic group selected from the group consisting of tetrahydrofuryl, dioxolanyl, furyl, thienyl, isoxazolyl, pyridyl, benzimidazolyl, benzothiazolyl, benzoxazolyl, benzopyranyl, quinolyl, isoquinolyl, tetrahydroisoquinolyl, benzothienyl and benzofuryl, each of which may have one or more suitable substituent(s), or a pharmaceutically acceptable salt thereof, which are useful as a medicament. |
申请公布号 |
WO9604254(A2) |
申请公布日期 |
1996.02.15 |
申请号 |
WO1995JP01497 |
申请日期 |
1995.07.27 |
申请人 |
FUJISAWA PHARMACEUTICAL CO., LTD.;NIPPON SHOKUBAI CO., LTD.;SATO, YOSHINARI;SAKANE, KAZUO;TABUCHI, SEIICHIRO;MITSUI, HITOSHI;KATSUMI, IKUYO;SATOH, YUICHI |
发明人 |
SATO, YOSHINARI;SAKANE, KAZUO;TABUCHI, SEIICHIRO;MITSUI, HITOSHI;KATSUMI, IKUYO;SATOH, YUICHI |
分类号 |
C07D243/14;A61K31/55;A61K31/551;A61P1/00;A61P25/04;A61P25/18;C07D243/24;C07D243/26;C07D401/06;C07D403/06;C07D405/06;C07D409/06;C07D413/06;C07D417/06;C07D487/08 |
主分类号 |
C07D243/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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