Novel fibrinogen receptor antagonists of the formula X-Y-Z-Aryl-A-B are provided in which the claimed compounds exhibit fibrinogen receptor antagonist activity, inhibit platelet aggregation and are therefore useful in modulating thrombus formation.
申请公布号
CA2150550(A1)
申请公布日期
1994.06.09
申请号
CA19932150550
申请日期
1993.11.29
申请人
MERCK & CO., INC.
发明人
EGBERTSON, MELISSA S.;TURCHI, LAURA M.;HARTMAN, GEORGE D.;HALCZENKO, WASYL;WHITMAN, DAVID B.;PERKINS, JAMES J.;KRAUSE, AMY E.;IHLE, NATHAN;CLAREMON, DAVID A.;HOFFMAN, WILLIAM;DUGGAN, MARK E.