Verfahren zur Herstellung von Salzen cyclischer Amidine
摘要
The invention relates to a method for producing salts of cyclic amidines of general formula (I). Known methods for producing salts of compound (I) only produce low yields. According to the invention, the appropriate omega -amino- alpha -amino acids are selectively protected in the omega -amino function. These protected compounds are decarboxylated oxidatively using halogen derivatives and the oxidatively decarboxylated substances are then cyclised with acid being added. This results in better yields of the salts of compound (I).
申请公布号
DE19754322(A1)
申请公布日期
1999.06.10
申请号
DE19971054322
申请日期
1997.12.08
申请人
DEGUSSA-HUELS AG, 45772 MARL, DE
发明人
MOST, DIETER, DR., 63486 BRUCHKOEBEL, DE;DRAUZ, KARLHEINZ, PROF. DR., 63579 FREIGERICHT, DE