发明名称 ACYL DERIVATIVES OF 5- (2-(4 -(1, 2 BENZISOTHIAZOLE -3- YL)-1- PIPERAZINYL) ETHYL)- 6-CHLORO -1, 3-DIHYDRO -2H -INDOL-2 -ONE HAVING NEUROLEPTIC ACTIVITY.
摘要 <p>A process for preparing acyl derivatives as prodrugs of 5- (2- (4- (1, 2 benzisothiazole- 3-yl)- 1-piperazinyl) ethyl-6 -chloro-1, 3-dihydro -2H- indol- 2- one and pharmaceutically acceptable acid addition salts and methods of use as an antipsychotic.</p>
申请公布号 MXPA05002734(A) 申请公布日期 2005.05.23
申请号 MX2005PA02734 申请日期 2003.10.13
申请人 PFIZER PRODUCTS INC. 发明人 COLON-CRUZ, ROBERTO
分类号 A61P25/18;C07D417/12;(IPC1-7):A61K31/428 主分类号 A61P25/18
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