发明名称 PARASITE CONTROL AGENT FOR PARASITICIDE
摘要 A parasite-control or parasiticide agent that exhibits excellent effects of controlling or expelling parasites, particularly endoparasites and that can be used safely contains at least one selected from the group consisting of compounds represented by formula (I) and salts thereof as an active ingredient thereof;;(In the formula (I), Cy represents a heteroaryl group or the like, X represents a halogeno group or the like, n is an integer of 0 to 5, in the case where n is 2 or more, X is identical or different, R1 represents an unsubstituted or substituted C1-6 alkyl group or the like, A represents a nitrogen atom or the like, R2, R3, and R4 each independently represents a hydrogen atom, an unsubstituted or substituted C1-6 alkyl group, or the like, and R5 represents an unsubstituted or substituted C6-10 aryl group, unsubstituted or substituted heteroaryl group, or the like.)
申请公布号 US2017035711(A1) 申请公布日期 2017.02.09
申请号 US201515304144 申请日期 2015.04.20
申请人 Nippon Soda Co., Ltd. 发明人 IWASA Takao
分类号 A61K31/17;A61K31/44;A61K31/505;A61K31/426;A61K31/506;A61K31/41;A61K31/444;A61K31/4965;A61K31/53;A61K31/4402;A61K31/4196 主分类号 A61K31/17
代理机构 代理人
主权项 1. A parasite-control or parasiticide agent comprising at least one selected from the group consisting of compounds represented by formula (I) and salts thereof as an active ingredient thereof:(in the formula (I), Cy represents a C6-10 aryl group or a heteroaryl group, X represents a halogeno group, an unsubstituted or substituted C1-6 alkyl group, an unsubstituted or substituted C3-8 cycloalkyl group, an unsubstituted or substituted C2-6 alkenyl group, an unsubstituted or substituted C2-6 alkynyl group, a hydroxyl group, an unsubstituted or substituted C1-6 alkoxy group, an unsubstituted or substituted amino group, an unsubstituted or substituted C1-7 acyl group, an unsubstituted or substituted C1-6 alkoxycarbonyl group, an unsubstituted or substituted C1-6 alkylaminocarbonyl group, an unsubstituted or substituted C1-6 alkylthio group, an unsubstituted or substituted C1-6 alkylsulfinyl group, an unsubstituted or substituted C1-6 alkylsulfonyl group, an unsubstituted or substituted C6-10 aryl group, an unsubstituted or substituted heteroaryl group, a nitro group, or a cyano group, n represents a number of X on Cy and is an integer of 0 to 5, and when n is 2 or more, X is identical or different, R1 represents an unsubstituted or substituted C1-6 alkyl group, an unsubstituted or substituted C2-6 alkenyl group, or an unsubstituted or substituted C2-6 alkynyl group, A represents a group represented by CR1a or a nitrogen atom (wherein R1a represents a hydrogen atom, an unsubstituted or substituted C1-6 alkyl group, an unsubstituted or substituted C2-6 alkenyl group, or an unsubstituted or substituted C2-6 alkynyl group), R2 represents a hydrogen atom, an unsubstituted or substituted C1-6 alkyl group, an unsubstituted or substituted C2-6 alkenyl group, an unsubstituted or substituted C2-6 alkynyl group, an unsubstituted or substituted C1-7 acyl group, or an unsubstituted or substituted C1-6 alkoxycarbonyl group, R3 and R4 each independently represents a hydrogen atom, an unsubstituted or substituted C1-6 alkyl group, an unsubstituted or substituted C2-6 alkenyl group, an unsubstituted or substituted C2-6 alkynyl group, or a cyano group, R5 represents an unsubstituted or substituted C1-6 alkyl group, an unsubstituted or substituted C2-6 alkenyl group, an unsubstituted or substituted C2-6 alkynyl group, an unsubstituted or substituted C1-7 acyl group, a carboxyl group, an unsubstituted or substituted C1-6 alkoxycarbonyl group, an unsubstituted or substituted C2-6 alkenyloxycarbonyl group, an unsubstituted or substituted C2-6 alkynyloxycarbonyl group, an aminocarbonyl group, an unsubstituted or substituted C1-6 alkylaminocarbonyl group, an unsubstituted or substituted C6-10 aryl group, or an unsubstituted or substituted heteroaryl group).
地址 Chiyoda-ku, Tokyo JP