发明名称 THIOPHENE OR THIAZOLE DERIVATIVES AND THEIR USE AS PI3K INHIBITORS
摘要 This invention provides compounds of formula (I) wherein R, R, CY, Y, Y, X, X, and Xare as described in the specification. The compounds are inhibitors of PI3K and are thus useful for treating proliferative, inflammatory, or cardiovascular disorders.
申请公布号 UA106206(C2) 申请公布日期 2014.08.11
申请号 UA20110000563 申请日期 2009.06.17
申请人 MILLENNIUM PHARMACEUTICALS, INC. 发明人 CARDIN, DAVID, P.;GAULIN, JEFFREY, L.;GREENSPAN, PAUL, D.;VYSKOCIL, STEPAN;XU, TIANLIN;RENOU, CHRISTELLE, C.
分类号 C07D409/04;A61K31/4196;A61K31/427;A61K31/5377;C07D409/14;C07D417/04 主分类号 C07D409/04
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