摘要 |
Compounds of the formula and pharmaceutically acceptable salts thereof, wherein X1, X2, X3, X4, X5, X6, X7, R1, and Q1 are defined herein, inhibit the IGF-1R enzyme and are useful for the treatment and/or prevention of hyperproliferative diseases such as cancer, inflammation, psoriasis, allergy/asthma, disease and conditions of the immune system, disease and conditions of the central nervous system. |
申请人 |
ARNOLD LEE D.;CESARIO CARA;COATE HEATHER;CREW ANDREW P.;DONG HANQING;FOREMAN KENNETH;HONDA AYAKO;LAUFER RADOSLAW;LI AN-HU;MULVIHILL KRISTEN MICHELLE;MULVIHILL MARK J.;NIGRO ANTHONY I.;PANICKER BIJOY;STEINIG ARNO G.;SUN YINGCHUAN;WENG QUINGHUA;WERNER DOUGLAS S.;WYLE MICHAEL J.;ZHANG TAO;OSI PHARMACEUTICALS, LLC |
发明人 |
ARNOLD LEE D.;CESARIO CARA;COATE HEATHER;CREW ANDREW P.;DONG HANQING;FOREMAN KENNETH;HONDA AYAKO;LAUFER RADOSLAW;LI AN-HU;MULVIHILL KRISTEN MICHELLE;MULVIHILL MARK J.;NIGRO ANTHONY I.;PANICKER BIJOY;STEINIG ARNO G.;SUN YINGCHUAN;WENG QUINGHUA;WERNER DOUGLAS S.;WYLE MICHAEL J.;ZHANG TAO |