发明名称 6,6-bicyclic ring substituted heterobicyclic protein kinase inhibitors
摘要 Compounds of the formula and pharmaceutically acceptable salts thereof, wherein X1, X2, X3, X4, X5, X6, X7, R1, and Q1 are defined herein, inhibit the IGF-1R enzyme and are useful for the treatment and/or prevention of hyperproliferative diseases such as cancer, inflammation, psoriasis, allergy/asthma, disease and conditions of the immune system, disease and conditions of the central nervous system.
申请公布号 US8735405(B2) 申请公布日期 2014.05.27
申请号 US201213446629 申请日期 2012.04.13
申请人 ARNOLD LEE D.;CESARIO CARA;COATE HEATHER;CREW ANDREW P.;DONG HANQING;FOREMAN KENNETH;HONDA AYAKO;LAUFER RADOSLAW;LI AN-HU;MULVIHILL KRISTEN MICHELLE;MULVIHILL MARK J.;NIGRO ANTHONY I.;PANICKER BIJOY;STEINIG ARNO G.;SUN YINGCHUAN;WENG QUINGHUA;WERNER DOUGLAS S.;WYLE MICHAEL J.;ZHANG TAO;OSI PHARMACEUTICALS, LLC 发明人 ARNOLD LEE D.;CESARIO CARA;COATE HEATHER;CREW ANDREW P.;DONG HANQING;FOREMAN KENNETH;HONDA AYAKO;LAUFER RADOSLAW;LI AN-HU;MULVIHILL KRISTEN MICHELLE;MULVIHILL MARK J.;NIGRO ANTHONY I.;PANICKER BIJOY;STEINIG ARNO G.;SUN YINGCHUAN;WENG QUINGHUA;WERNER DOUGLAS S.;WYLE MICHAEL J.;ZHANG TAO
分类号 A01N43/90;A61K31/437;A61K31/4985;A61K31/5025;A61K31/519;A61K31/53;C07D471/04;C07D487/00;C07D487/04 主分类号 A01N43/90
代理机构 代理人
主权项
地址