| 发明名称 |
NOVEL PYRAZOLE AND IMIDAZOLE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS |
| 摘要 |
<p>The present invention relates to pyrazole and imidazole derivatives of formula (I) wherein U, V, L, X, Y, R1, (R2)n and (R3)m and ring A are as described in the description, to their preparation, to pharmaceutically acceptable salts thereof, and to their use as pharmaceuticals, to pharmaceutical compositions containing one or more compounds of formula (I), and especially to their use as orexin receptor antagonists.</p> |
| 申请公布号 |
EP2675801(A1) |
申请公布日期 |
2013.12.25 |
| 申请号 |
EP20120709375 |
申请日期 |
2012.02.17 |
| 申请人 |
ACTELION PHARMACEUTICALS LTD. |
发明人 |
BOLLI, MARTIN;BOSS, CHRISTOPH;BROTSCHI, CHRISTINE;GUDE, MARKUS;HEIDMANN, BIBIA;SIFFERLEN, THIERRY;WILLIAMS, JODI,T. |
| 分类号 |
C07D413/12;A61K31/4155;A61K31/4178;A61K31/422;A61P25/00;C07D413/14;C07D417/12;C07D417/14 |
主分类号 |
C07D413/12 |
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