发明名称 |
Solid Forms of (R)-1(2,2-Difluorobenzo[D][1,3]Dioxol-5-yl)-N-(1-(2,3-Dihydroxypropyl-6-Fluoro-2-(1-Hydroxy-2-Methylpropan-2-yl)-1H-Indol-5-yl)-Cyclopropanecarboxamide |
摘要 |
The present invention relates to solid forms of (R)-1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)-N-(1-(2,3-dihydroxypropyl)-6-fluoro-2-(1-hydroxy-2-methylpropan-2-yl)-1H-indol-5-yl)cyclopropanecarboxamide (Compound 1) in substantially crystalline form (Form A) or amorphous form, pharmaceutical compositions thereof, and methods of treatment therewith.
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申请公布号 |
US2013143918(A1) |
申请公布日期 |
2013.06.06 |
申请号 |
US201213624241 |
申请日期 |
2012.09.21 |
申请人 |
VERTEX PHARMACEUTICALS INCORPORATED;VERTEX PHARMACEUTICALS INCORPORATED |
发明人 |
KESHAVARZ-SHOKRI ALI;ZHANG BEILI;ALCACIO TIM EDWARD;LEE ELAINE CHUNGMIN;ZHANG YUEGANG;KRAWIEC MARIUSZ |
分类号 |
A61K31/404;A61K31/47;A61K45/06;C07D405/12;C07D495/04 |
主分类号 |
A61K31/404 |
代理机构 |
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地址 |
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