发明名称 FUSED BICYCLIC DERIVATIVES OF 2,4-DIAMINOPYRIMIDINE AS ALK AND C-MET INHIBITORS
摘要 <p>The present invention provides a compound of formula I or II or a pharmaceutically acceptable salt form thereof, wherein R<SUP>1</SUP>, R<SUP>2</SUP>, R<SUP>3</SUP>, R<SUP>4</SUP>, R<SUP>5</SUP>, A<SUP>1</SUP>, A<SUP>2</SUP>, A<SUP>3</SUP>, A<SUP>4</SUP>, and A<SUP>5</SUP>, are as defined herein. The compounds of formula I or II have ALK and/or c-Met inhibitory activity, and may be used to treat proliferative disorders.</p>
申请公布号 WO2008051547(A1) 申请公布日期 2008.05.02
申请号 WO2007US22496 申请日期 2007.10.23
申请人 CEPHALON, INC.;PHARMACOPEIA DRUG DISCOVERY, INC.;AHMED, GULZAR;BOHNSTEDT, ADOLPH;BRESLIN, HENRY, JOSEPH;BURKE, JASON;CURRY, MATTHEW, A.;DIEBOLD, JAMES, L.;DORSEY, BRUCE;DUGAN, BENJAMIN, J.;FENG, DAMING;GINGRICH, DIANE, E.;GUO, TAO;HO, KOC-KAN;LEARN, KEITH, S.;LISKO, JOSEPH, G.;LIU, RONG-QIANG;MESAROS, EUGEN, F.;MILKIEWICZ, KAREN;OTT, GREGORY, R.;PARRISH, JONATHAN;THEROFF, JAY, P.;THIEU, THO, V.;TRIPATHY, RABINDRANATH;UNDERINER, THEODORE, L.;WAGNER, JASON, C.;WEINBERG, LINDA;WELLS, GREGORY, J.;YOU, MING;ZIFICSAK, CRAIG, A. 发明人 AHMED, GULZAR;BOHNSTEDT, ADOLPH;BRESLIN, HENRY, JOSEPH;BURKE, JASON;CURRY, MATTHEW, A.;DIEBOLD, JAMES, L.;DORSEY, BRUCE;DUGAN, BENJAMIN, J.;FENG, DAMING;GINGRICH, DIANE, E.;GUO, TAO;HO, KOC-KAN;LEARN, KEITH, S.;LISKO, JOSEPH, G.;LIU, RONG-QIANG;MESAROS, EUGEN, F.;MILKIEWICZ, KAREN;OTT, GREGORY, R.;PARRISH, JONATHAN;THEROFF, JAY, P.;THIEU, THO, V.;TRIPATHY, RABINDRANATH;UNDERINER, THEODORE, L.;WAGNER, JASON, C.;WEINBERG, LINDA;WELLS, GREGORY, J.;YOU, MING;ZIFICSAK, CRAIG, A.
分类号 C07D239/48;A61K31/495;A61P35/00;C07D403/12;C07D403/14;C07D405/12;C07D405/14;C07D413/12;C07D417/12;C07D417/14 主分类号 C07D239/48
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