发明名称 CRYSTALLINE SOLVATES AND COMPLEXES OF (IS) -1, 5-ANHYDRO-L-C- (3- ( (PHENYL) METHYL) PHENYL) -D-GLUCITOL DERIVATIVES WITH AMINO ACIDS AS SGLT2 INHIBITORS FOR THE TREATMENT OF DIABETES
摘要 The present invention relates to physical crystal structures of a compound of the formula I: wherein R1, R2, R2a, R3 and R4 are as defined herein, especially pharmaceutical compositions containing structures of compound I or II, processes for preparing same, intermediates used in preparing same, and methods of treating diseases such as diabetes using such structures.
申请公布号 WO2008002824(A1) 申请公布日期 2008.01.03
申请号 WO2007US71749 申请日期 2007.06.21
申请人 BRISTOL-MYERS SQUIBB COMPANY;GOUGOUTAS, JACK, Z.;LOBINGER, HILDEGARD;RAMAKRISHNAN, SRIVIDYA;DESHPANDE, PRASHANT, P.;BIEN, JEFFREY, T.;LAI, CHIAJEN;WANG, CHENCHI;RIEBEL, PETER;GROSSO, JOHN, ANTHONY;NIRSCHL, ALEXANDRA, A.;SINGH, JANAK;DIMARCO, JOHN, D. 发明人 GOUGOUTAS, JACK, Z.;LOBINGER, HILDEGARD;RAMAKRISHNAN, SRIVIDYA;DESHPANDE, PRASHANT, P.;BIEN, JEFFREY, T.;LAI, CHIAJEN;WANG, CHENCHI;RIEBEL, PETER;GROSSO, JOHN, ANTHONY;NIRSCHL, ALEXANDRA, A.;SINGH, JANAK;DIMARCO, JOHN, D.
分类号 C07H7/04;A61K31/70;A61P3/10 主分类号 C07H7/04
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