发明名称 |
Process for the preparation of a boron-substituted porphyrin |
摘要 |
Processes are disclosed for the preparation of a compound having the formula: (I) and intermediate compounds wherein M is a single-photon-emission tomography imageable radiometal and/or a paramagnetic metal, R is hydrogen or a halogen provided that at least one R is halogen and Y is selected from ortho, meta or para O(CH2)nC2HB9H10 or O(CH2)nC2HB10H10 wherein n is 0 or an integer from 1 to 20 and O(CH2)nC2HB9H10 is nido ortho-, meta- or para-carborane and O(CH2)nC2HB10H10 is ortho-, meta- or para-carborane. |
申请公布号 |
GB2436767(A) |
申请公布日期 |
2007.10.03 |
申请号 |
GB20070013798 |
申请日期 |
2007.07.16 |
申请人 |
PSIMEI PHARMACEUTICALS PLC |
发明人 |
KE-DONG LI;ANTHONY DAVID BENTHAM;BIPIN CHANDRA MULJIBHAI PATEL |
分类号 |
C07D487/22;A61K41/00;A61P35/00;C07F5/05 |
主分类号 |
C07D487/22 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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