发明名称 |
AMIDINODERIVAT AV MITOMYCIN-C OCH FORFARANDE FOR FRAMSTELLNING DERAV |
摘要 |
Mitomycin A, mitomycin C, and porfiromycin react with amide acetals and other amide derivatives to produce amidine derivatives having antitumor activity against experimental animal tumors. The amidines derived from mitomycin C are useful intermediates in reactions with primary amines to produce both known and novel 7-amino-9a-methoxymitosanes having antitumor activity against experimental animal tumors. |
申请公布号 |
SE455504(B) |
申请公布日期 |
1988.07.18 |
申请号 |
SE19830003160 |
申请日期 |
1983.06.03 |
申请人 |
BRISTOL-MYERS COMPANY |
发明人 |
D M * VYAS;T * KANEKO;T W * DOYLE |
分类号 |
C07D487/14;(IPC1-7):C07D487/14 |
主分类号 |
C07D487/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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