发明名称 DIKLORANILINDERIVAT
摘要 The invention provides compounds of the general formula (I) <IMAGE> (I) wherein X represents a bond or a C1-6 alkylene, C2-6 alkenylene or C2-6 alkynylene chain, and Y represents a bond, or a C1-4 alkylene, C2-4 alkenylene or C2-4 alkynylene chain with the proviso that the sum total of carbon atoms in X and Y is not more than 8; Py represents a pyridyl group optionally substituted by one or two substituents selected from halogen atoms, hydroxy, C1-3 alkyl and C1-3 alkoxy groups; and R1 and R2 each represent a hydrogen atom or a C1-3 alkyl group, with the proviso that the sum total of carbon atoms in R1 and R2 is not more than 4; and physiologically acceptable salts and solvates (e.g. hydrates) thereof. The compounds have a stimulant action at beta 2-adrenoreceptors and may be used in the treatment of diseases associated with reversible airways obstruction such as asthma and chronic bronchitis.
申请公布号 SE8700535(D0) 申请公布日期 1987.02.11
申请号 SE19870000535 申请日期 1987.02.11
申请人 GLAXO GROUP LTD 发明人 L H C * LUNTS
分类号 C07D213/38;A61K31/44;A61K31/4402;A61K31/4406;A61K31/4409;A61K31/4418;A61K31/4425;A61P1/04;A61P11/00;A61P11/08;A61P13/02;A61P15/00;A61P25/24;A61P25/26;A61P27/02;A61P27/14;A61P29/00;A61P37/08;C07D213/30;C07D213/61;C07D213/63;C07D213/65;(IPC1-7):C07D/ 主分类号 C07D213/38
代理机构 代理人
主权项
地址